Antimalarial Activity of C-10 Substituted Triazolyl Artemisinin
نویسندگان
چکیده
منابع مشابه
Antimalarial Activity of C-10 Substituted Triazolyl Artemisinin
We synthesized C-10 substituted triazolyl artemisinins by the Huisgen cycloaddition reaction between dihydroartemisinins (2) and variously substituted 1, 2, 3-triazoles (8a-8h). The antimalarial activities of 32 novel artemisinin derivatives were screened against a chloroquine-resistant parasite. Among them, triazolyl artemisinins with electron-withdrawing groups showed stronger antimalarial ac...
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ژورنال
عنوان ژورنال: The Korean Journal of Parasitology
سال: 2017
ISSN: 0023-4001,1738-0006
DOI: 10.3347/kjp.2017.55.6.661